Palladium(II)-catalyzed othro-C-H-benzoxylation of 2-arylpyridines by oxidative coupling with aryl acylperoxides.
نویسندگان
چکیده
A palladium(II)-catalyzed ortho-benzoxylation of 2-arylpyridines with aryl acylperoxides was developed. With pyridyl as directing group, the benzoxylation reaction exhibits remarkable regioselectivity and excellent functional group tolerance, providing the products in up to 87% yield.
منابع مشابه
Copper(II)-catalyzed ortho-functionalization of 2-arylpyridines with acyl chlorides.
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ورودعنوان ژورنال:
- Molecules
دوره 18 4 شماره
صفحات -
تاریخ انتشار 2013